GR 103691( —— )

Catalog No. M23720 CAS No. 162408-66-4

GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).?

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

GR 103691
Note

Research use only, not for human use.
Brief Description

GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).?
Description

GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).?It shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites.
In Vitro

GR 103691 shows marked affinity for serotonin1A (5-HT1A) receptors (Ki of 5.8 nM) and α-1 adrenoceptors (Ki of 12.6 nM).
In Vivo

——
Synonyms

——
Pathway

GPCR/G Protein
Target

Dopamine Receptor
Recptor

D3
Research Area

——
Indication

——

Chemical Information

CAS Number

162408-66-4
Formula Weight

485.62
Molecular Formula

C30H35N3O3
Purity

>98% (HPLC)
Solubility

DMSO:10 mM
SMILES

O=C(C1=CC=C(C2=CC=C(C(C)=O)C=C2)C=C1)NCCCCN3CCN(C4=CC=CC=C4OC)CC3
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Audinot V, et al. A comparative in vitro and in vivo pharmacological characterization of the novel dopamine D3 receptor antagonists (+)-S 14297, nafadotride, GR 103,691 and U 99194. J Pharmacol Exp Ther. 1998 Oct;287(1):187-97.

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